1: With trichlorophosphate in N,N-dimethyl-formamide T=20 - 80°C; 0.25 h; 2: With sodium hydroxide; water in N,N-dimethyl-formamide 3: With hydrogenchloride; water T=70°C; 0.5 h;
参考文献
TargeGen, Inc.
Patent: US2007/259876 A1, 2007 ;
Location in patent: Page/Page column 18 ;
US 20070259876 A1