5,6-二氟-1H-吲哚-3-甲醛合成路线 (共 2 条)
反应条件
1: N,N-dimethyl-formamide With trichlorophosphate T=0 - 20°C; 1.5 h; 2: 5,6-difluoroindole in N,N-dimethyl-formamide T=0 - 20°C; 15.5 h;
参考文献
Bayer Schering Pharma Aktiengesellschaft
Patent: EP1932831 A1, 2008 ;
Location in patent: Page/Page column 45 ;
参考文献
Vernalis Research Limited
Patent: US6433175 B1, 2002 ;