4-甲基-2-(三氟乙酰基)环己酮合成路线 (共 1 条)
反应条件
1: (RS)-4-methylcyclohexanone With lithium diisopropyl amide in tetrahydrofuran T=-70°C; 0.416667 h; 2: ethyl-α,α,α-trifluoroacetate in tetrahydrofuran T=-70 - 20°C; 2.16667 h;
参考文献
GLAXO GROUP LIMITED
Patent: WO2008/148832 A1, 2008 ;
Location in patent: Page/Page column 34-35 ;
WO 2008/148832 A1