1H-1,2,3-噻唑并[4,5-c]吡啶合成路线 （共 12 条）
反应条件
1: N-(3-aminopyridin-4-yl)acetamide With NOBF4 in acetonitrile T=0°C; 0.333333 h; 2: isopropylamine in acetonitrile T=20°C;
参考文献
Holt, Jarle; Fiksdahl, Anne
Journal of Heterocyclic Chemistry, 2006 , vol. 43, # 2 p. 417 - 423
反应条件
1: 3-amino-4-pyridylcarbamic acid methyl ester With NOBF4 in acetonitrile T=0°C; 0.333333 h; 2: isopropylamine in acetonitrile T=20°C;
参考文献
Holt, Jarle; Fiksdahl, Anne
Journal of Heterocyclic Chemistry, 2006 , vol. 43, # 2 p. 417 - 423
反应条件
1: 3-amino-4-pyridylcarbamic acid methyl ester With NOBF4 in acetonitrile T=0°C; 0.333333 h; 2: benzylamine in acetonitrile T=20°C;
参考文献
Holt, Jarle; Fiksdahl, Anne
Journal of Heterocyclic Chemistry, 2006 , vol. 43, # 2 p. 417 - 423
反应条件
acetic acid; sodium nitrite T=10 - 25°C; 1 h;
参考文献
Balachari, Devan; Trudell, Mark L.
Tetrahedron Letters, 1997 , vol. 38, # 50 p. 8607 - 8610
反应条件
1: 3-amino-4-pyridinylcarbamic acid ethyl ester With NOBF4 in acetonitrile T=0°C; 0.333333 h; 2: isopropylamine in acetonitrile T=20°C;
参考文献
Holt, Jarle; Fiksdahl, Anne
Journal of Heterocyclic Chemistry, 2006 , vol. 43, # 2 p. 417 - 423
反应条件
1: (3-Amino-pyridin-4-yl)-carbamic acid tert-butyl ester With NOBF4 in acetonitrile T=0°C; 0.333333 h; 2: isopropylamine in acetonitrile T=20°C;
参考文献
Holt, Jarle; Fiksdahl, Anne
Journal of Heterocyclic Chemistry, 2006 , vol. 43, # 2 p. 417 - 423
反应条件
1: N-(3-aminopyridin-4-yl)benzamide With NOBF4 in acetonitrile T=0°C; 0.333333 h; 2: isopropylamine in acetonitrile T=20°C;
参考文献
Holt, Jarle; Fiksdahl, Anne
Journal of Heterocyclic Chemistry, 2006 , vol. 43, # 2 p. 417 - 423
反应条件
1: 3-amino-4-pyridinylcarbamic acid ethyl ester With NOBF4 in acetonitrile T=0°C; 0.333333 h; 2: benzylamine in acetonitrile T=20°C;
参考文献
Holt, Jarle; Fiksdahl, Anne
Journal of Heterocyclic Chemistry, 2006 , vol. 43, # 2 p. 417 - 423
反应条件
1: N-(3-aminopyridin-4-yl)acetamide With NOBF4 in acetonitrile T=0°C; 0.333333 h; 2: benzylamine in acetonitrile T=20°C;
参考文献
Holt, Jarle; Fiksdahl, Anne
Journal of Heterocyclic Chemistry, 2006 , vol. 43, # 2 p. 417 - 423
反应条件
1: (3-Amino-pyridin-4-yl)-carbamic acid tert-butyl ester With NOBF4 in acetonitrile T=0°C; 0.333333 h; 2: benzylamine in acetonitrile T=20°C;
参考文献
Holt, Jarle; Fiksdahl, Anne
Journal of Heterocyclic Chemistry, 2006 , vol. 43, # 2 p. 417 - 423
