咪唑并[1,5-a]吡啶合成路线 （共 16 条）
反应条件
palladium diacetate; acetic acid; silver carbonate in dimethyl sulfoxide; N,N-dimethyl-formamide T=120°C; 0.833333 h; Inert atmosphere;
参考文献
Journal of Organic Chemistry, , vol. 77, # 12 p. 5381 - 5388
反应条件
N-bromosuccinmide in dichloromethane
T=-78 - 20°C; 1.5 h; Inert atmosphere;
参考文献
Shibahara, Fumitoshi; Dohke, Yoshimasa; Murai, Toshiaki
Journal of Organic Chemistry, 2012 , vol. 77, # 12 p. 5381 - 5388
反应条件
N-bromosuccinmide in dichloromethane
T=-78 - 20°C; 1.5 h; Inert atmosphere;
参考文献
Shibahara, Fumitoshi; Dohke, Yoshimasa; Murai, Toshiaki
Journal of Organic Chemistry, 2012 , vol. 77, # 12 p. 5381 - 5388
反应条件
palladium diacetate; acetic acid; silver carbonate in dimethyl sulfoxide; N,N-dimethyl-formamide
T=120°C; 0.833333 h; Inert atmosphere;
参考文献
Shibahara, Fumitoshi; Dohke, Yoshimasa; Murai, Toshiaki
Journal of Organic Chemistry, 2012 , vol. 77, # 12 p. 5381 - 5388
反应条件
palladium diacetate; acetic acid; silver carbonate in dimethyl sulfoxide; N,N-dimethyl-formamide
T=120°C; 0.833333 h; Inert atmosphere;
参考文献
Shibahara, Fumitoshi; Dohke, Yoshimasa; Murai, Toshiaki
Journal of Organic Chemistry, 2012 , vol. 77, # 12 p. 5381 - 5388
反应条件
1: With hydrogen; trifluoroacetic acid; platinum(IV) oxide
T=20°C;
2: With sodium hydroxide
参考文献
MILLENNIUM PHARMACEUTICALS, INC.
Patent: WO2009/67233 A1, 2009 ;
Location in patent: Page/Page column 41 ;
