反应条件
1: 95 percent / 4 h / 0 - 20 °C
2: 1.) POCl3, Et3N, 2.) aq. Na2CO3 / 1.) CH2Cl2, 0 deg C, 1 h, 2.) CH2Cl2, 1 h
View Scheme
参考文献
Jacobsen, E. Jon; Stelzer, Lindsay S.; Belonga, Kenneth L.; Carter, Donald B.; Im, Wha Bin; Sethy, Vimala H.; Tang, Andrew H.; Von Voigtlander, Philip F.; Petke, James D.
Journal of Medicinal Chemistry, 1996 , vol. 39, # 19 p. 3820 - 3836