反应条件
1: 4-quinolynylmethyl 4-bromobenzoate With ammonium formate; 1,2-bis-(diphenylphosphino)ethane; bis(dibenzylideneacetone)-palladium(0) in dimethyl sulfoxide T=50°C; Reduction; Deprotection; 12 h; 2: methyl iodide With sodium carbonate in water; dimethyl sulfoxide T=20°C; Methylation; 12 h;
参考文献
Boutros, Andre; Legros, Jean-Yves; Fiaud, Jean-Claude
Tetrahedron, 2000 , vol. 56, # 15 p. 2239 - 2246