反应条件
1: (1S,2S,3R,5S)-3-(7-hydroxy-5-(propylthio)-3H-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)-5-(2-hydroxyethoxy)cyclopentane-1,2-diol With O-(6-chloro-1H-benzotriazol-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate; N-ethyl-N,N-diisopropylamine in N,N-dimethyl-formamide T=25°C; 0.25 h; Inert atmosphere; 2: (1R,2S)-2-(3,4-difluorophenyl)cyclopropanamine hydrochloride in N,N-dimethyl-formamide T=25°C; 16 h; Inert atmosphere;