[1,2,5]恶二唑并[3,4-b]吡啶 1-氧化物合成路线 （共 10 条）
反应条件
[bis(acetoxy)iodo]benzene in benzene T=60°C; 2 h;
参考文献
Binder, Dieter; Noe, Christian R.; Nussbaumer, Johannes; Prager, Bernhard C.
Monatshefte fuer Chemie, 1980 , vol. 111, p. 407 - 412
反应条件
1: 0.27 g / NaN3, 10percent HCl / aq. ethanol / 48 h / Heating 2: 0.27 g / toluene / 4 h / Heating View Scheme
参考文献
Boyer et al.
Journal of the American Chemical Society, 1953 , vol. 75, p. 5298
反应条件
in acetone T=-40.15°C; Rearrangement; Equilibrium constant;
参考文献
Cmoch; Kamienski; Kamienska-Trela; Stefaniak; Webb
Journal of Physical Organic Chemistry, 2000 , vol. 13, # 8 p. 480 - 488
反应条件
in acetone T=-40.15°C; Rearrangement; Equilibrium constant;
参考文献
Cmoch; Kamienski; Kamienska-Trela; Stefaniak; Webb
Journal of Physical Organic Chemistry, 2000 , vol. 13, # 8 p. 480 - 488
反应条件
dihydrogen peroxide in various solvent(s) 24 h; Ambient temperature; Yield given;
参考文献
Lowe-Ma, Charlotte K.; Nissan, Robin A.; Wilson, William S.
Journal of Organic Chemistry, 1990 , vol. 55, p. 3755 - 3761
反应条件
1: 20 percent / NH3 / methanol / 0.33 h / Heating
2: 27 percent / KOH, H2 / Raney-Ni W6 / ethanol; H2O
View Scheme
参考文献
Binder, Dieter; Noe, Christian R.; Nussbaumer, Johannes; Prager, Bernhard C.
Monatshefte fuer Chemie, 1980 , vol. 111, p. 407 - 412
反应条件
morpholine in acetone
参考文献
Binder; Georgopoulos; Noe; Nussbaumer; Prager; Turnowsky
Arzneimittel-Forschung/Drug Research, 1982 , vol. 32, # 1 p. 10 - 14
反应条件
ammonia in methanol; butanone
参考文献
Binder, Dieter; Noe, Christian R.; Nussbaumer, Johannes; Prager, Bernhard C.
Monatshefte fuer Chemie, 1980 , vol. 111, p. 407 - 412
反应条件
pyrrolidine in chloroform
15 h; Ambient temperature;
参考文献
Binder; Georgopoulos; Noe; Nussbaumer; Prager; Turnowsky
Arzneimittel-Forschung/Drug Research, 1982 , vol. 32, # 1 p. 10 - 14
参考文献
Binder, Dieter; Noe, Christian R.; Nussbaumer, Johannes; Prager, Bernhard C.
Monatshefte fuer Chemie, 1980 , vol. 111, p. 407 - 412
