4-(8-氟-3,4,5,6-四氢-6-氧代-1H-氮杂卓并[5,4,3-cd]吲哚-2-基)苯甲醛合成路线 (共 2 条)
反应条件
1: hydrogenchloride; sodium cyanoborohydride / methanol; water; tetrahydrofuran; ethanol / |Large scale 2: sodium hydroxide / methanol; water; tetrahydrofuran / 18 h / 20 °C / |Large scale View Scheme
参考文献
Organic Process Research and Development, , vol. 16, # 12 p. 1897 - 1904