反应条件
1: 63 percent / Et3N, 4-(dimethylamino)pyridine / CH2Cl2 / 24 h / Heating 2: 55 percent / conc. H2SO4, conc. HNO3 / -5 °C View Scheme
参考文献
Munk, Stephen A.; Harcourt, Dale; Ambrus, Gyoergy; Denys, Lydia; Gluchowski, Charles; Burke, James A.; Kharlamb, Alexander B.; Manlapaz, Cynthia A.; Padillo, Edwin U.; Runde, Eileen; Williams, Linda; Wheeler, Larry A.; Garst, Michael E.
Journal of Medicinal Chemistry, 1996 , vol. 39, # 18 p. 3533 - 3538