2-(3-氨基苯基)-1-吗啉-4-基-乙酮合成路线 (共 2 条)
反应条件
1: 55 percent / Et3N, EDC, DMAP 2: H2 / 10percent Pd/C / ethyl acetate / 1.5 h View Scheme
参考文献
Collins, Jon L.; Shearer, Barry G.; Oplinger, Jeffrey A.; Lee, Shuliang; Garvey, Edward P.; Salter, Mark; Duffy, Claire; Burnette, Thimysta C.; Furfine, Eric S.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 15 p. 2858 - 2871
参考文献
Deciphera Pharmaceuticals, LLC
Patent: US7666895 B2, 2010 ;