4-氟-5-甲氧基-1H-吲哚合成路线 （共 3 条）
反应条件
copper(l) iodide in ethyl acetate T=140°C; 5 h;
参考文献
Laban, Uros; Kurrasch-Orbaugh, Deborah; Marona-Lewicka, Danuta; E. Nichols, David
Bioorganic and Medicinal Chemistry Letters, 2001 , vol. 11, # 6 p. 793 - 795
参考文献
NYCOMED GMBH
Patent: WO2007/96395 A1, 2007 ;
Location in patent: Page/Page column 124-125 ;
反应条件
1: NaHSO3 / 24 h / 20 °C 2: 3 h / Heating 3: aq. Br2 / 0 °C 4: 5 N aq. NaOH 5: 70 percent / CuI / ethyl acetate / 5 h / 140 °C View Scheme
参考文献
Laban, Uros; Kurrasch-Orbaugh, Deborah; Marona-Lewicka, Danuta; E. Nichols, David
Bioorganic and Medicinal Chemistry Letters, 2001 , vol. 11, # 6 p. 793 - 795
