反应条件
1: pyridine / 18 h / Ambient temperature 2: 1.) K2CO3 / 1.) DMF, 120 deg C, 1 h, 2.) DMF, 120 deg C 3: HCl, MeOH / Ambient temperature View Scheme
参考文献
Cavallaro, Rosaria A.; Filocamo, Luigi; Galuppi, Annamaria; Galione, Antony; Brufani, Mario; Genazzani, Armando A.
Journal of Medicinal Chemistry, 1999 , vol. 42, # 14 p. 2527 - 2534