四唑并[1,5-a]喹喔啉-4-醇合成路线 (共 5 条)
参考文献
Eli Lilly and Company
Patent: US5153196 A1, 1992 ;
US 5153196 A
反应条件
dihydrogen peroxide; acetic acid T=85°C; 16 h;
参考文献
McQuaid; Smith; South; Mitch; Schoepp; True; Calligaro; O'Malley; Lodge; Ornstein
Journal of Medicinal Chemistry, 1992 , vol. 35, # 18 p. 3319 - 3324
反应条件
1: sodium azide / ethanol / 17 h / Heating 2: AcOH, 30 percent H2O2 / 16 h / 85 °C View Scheme
参考文献
McQuaid; Smith; South; Mitch; Schoepp; True; Calligaro; O'Malley; Lodge; Ornstein
Journal of Medicinal Chemistry, 1992 , vol. 35, # 18 p. 3319 - 3324
反应条件
potassium carbonate; sodium iodide in neat (no solvent)
1 h; Heating;
参考文献
Klicnar, Jiri; Toman, Jaromir
Collection of Czechoslovak Chemical Communications, 1981 , vol. 46, # 9 p. 2110 - 2115
参考文献
Deshmukh; Mali; Jadhav; Suryawanshi
Indian Journal of Chemistry - Section B Organic and Medicinal Chemistry, 2007 , vol. 46, # 7 p. 1211 - 1213