5-溴-2-氟苯胺合成路线

364-76-14-氟-3-硝基苯胺

2924-09-65-溴-2-氟苯胺

参考文献

Helvetica Chimica Acta, , vol. 66, # 1 p. 68 - 75

2924-09-65-溴-2-氟苯胺+

140-89-6乙基黄原酸钾

71216-20-15-溴-2-巯基苯并噻唑

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NOVO NORDISK A/S
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WO 2007/110364 A1

110-52-11,4-二溴丁烷+

2924-09-65-溴-2-氟苯胺

1280786-82-41-(5-溴-2-氟苯基)吡咯烷

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TREVENTIS CORPORATION; REED, Mark, A.; YADAV, Arun; BANFIELD, Scott, C.; BARDEN, Christopher, J.
Patent: WO2012/119035 A1, 2012 ;
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2924-09-65-溴-2-氟苯胺+

73183-34-3联硼酸频那醇酯

1003575-43-63-氨基-4-氟苯硼酸频那醇酯

参考文献

SELEXAGEN THERAPEUTICS, INC.; VERNIER, Jean-michel; HOPKINS, Stephanie; BOUNAUD, Pierre-Yves; O'CONNOR, Patrick; MATTHEWS, David; BENDER, Steve
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WO 2012/125981 A2

2924-09-65-溴-2-氟苯胺+

56-81-5甘油

1133115-78-25-溴-8-氟喹啉

参考文献

MERCK SHARP andamp; DOHME CORP.; LIN, Songnian; STEVENSON, Christian, P.; PARMEE, Emma, R.; XU, Libo; LIAO, Xibin; METZGER, Edward; LIANG, Rui; ZHANG, Fengqi; STELMACH, John, E.
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WO 2010/030722 A1

2924-09-65-溴-2-氟苯胺+

107-02-8丙烯醛

1133115-78-25-溴-8-氟喹啉

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GLAXO GROUP LIMITED; GORE, Paul Martin; HANCOCK, Ashley, Paul; HODGSON, Simon Teanby
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WO 2010/094643 A1

116272-41-42-碘-4-溴氟苯

参考文献

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2924-09-65-溴-2-氟苯胺

121-57-3对氨基苯磺酸

参考文献

Courtin, Alfred
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2924-09-65-溴-2-氟苯胺+

108-24-7乙酸酐

88288-12-4N-乙酰基-5-溴-2-氟苯胺

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GLAXO GROUP LIMITED
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