2-氟-4-碘苯胺合成路线

Katamreddy, Subba R.; Carpenter, Andrew J.; Ammala, Carina E.; Boros, Eric E.; Brashear, Ron L.; Briscoe, Celia P.; Bullard, Sarah R.; Caldwell, Richard D.; Conlee, Christopher R.; Croom, Dallas K.; Hart, Shane M.; Heyer, Dennis O.; Johnson, Paul R.; Kashatus, Jennifer A.; Minick, Doug J.; Peckham, Gregory E.; Ross, Sean A.; Roller, Shane G.; Samano, Vicente A.; Sauls, Howard R.; Tadepalli, Sarva M.; Thompson, James B.; Xu, Yun; Way, James M.
Journal of Medicinal Chemistry, 2012 , vol. 55, # 24 p. 10972 - 10994

314-41-02,3,4,6-四氟硝基苯+

29632-74-42-氟-4-碘苯胺

765962-71-8

参考文献

ARDEA BIOSCIENCES
Patent: US2007/238710 A1, 2007 ;
Location in patent: Page/Page column 46 ;
US 20070238710 A1

29632-74-42-氟-4-碘苯胺

85117-88-0N-(4-乙酰基-2-氟苯基)-乙胺

参考文献

Kruger; Keck; Noll; Pieper
Arzneimittel-Forschung/Drug Research, 1984 , vol. 34, # 11 A p. 1612 - 1624

6270-63-92-羟基吡嗪+

29632-74-42-氟-4-碘苯胺

863015-77-4

参考文献

Filipski, Kevin J.; Kohrt, Jeffrey T.; Casimiro-Garcia, Agustin; Van Huis, Chad A.; Dudley, Danette A.; Cody, Wayne L.; Bigge, Christopher F.; Desiraju, Shrilakshmi; Sun, Shaoyi; Maiti, Samarendra N.; Jaber, Mohamad R.; Edmunds, Jeremy J.
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148-24-3+

53406-38-5

863015-77-4

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Aventis Pharma Deutschland GmbH
Patent: EP1571154 A1, 2005 ;

29632-74-42-氟-4-碘苯胺+

393-53-33-氟吡啶-4-甲酸

885588-03-4

参考文献

MERCK SERONO S.A.; GOUTOPOULOS, Andreas; YU, Henry; ASKEW, Benny, C.; LIU-BUJALSKI, Lesley
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