反应条件
1: sodium hydride / N,N-dimethyl-formamide / 60 °C 2: [bis(acetoxy)iodo]benzene; 2,2,6,6-tetramethyl-1-piperidinyloxy, free radical / water; acetonitrile / 20 °C View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 23, # 1 p. 310 - 317