反应条件
1: 5-hydroxypyridine-2-carboxylic acid methyl ester With sodium hydride in N,N-dimethyl-formamide 0.5 h; 2: methyl iodide in N,N-dimethyl-formamide 1 h;
参考文献
Brewster, William Kirkland; Klittich, Carla Jean Rasmussen; Balko, Terry William; Breaux, Nneka Tuere; Erickson, William Randal; Hunter, James Edward; Lowe, Christian Thomas; Ricks, Michael John; Siddall, Thomas Lyman; Yerkes, Carla Nanette; Zhu, Yuanming
Patent: US2006/89370 A1, 2006 ;
Location in patent: Page/Page column 33 ;