5-氨基-1-Boc-苯并咪唑合成路线 （共 2 条）
反应条件
1: 1H-Benzoimidazol-5-ylamine With sodium hydride in DMF (N,N-dimethyl-formamide)
T=20°C; 1 h;
2: di-tert-butyl dicarbonate in DMF (N,N-dimethyl-formamide)
T=0 - 20°C; 18 h;
参考文献
Glaxo Wellcome Inc.
Patent: US6350747 B1, 2002 ;
Location in patent: Page column 50-51 ;
反应条件
palladium 10 on activated carbon; hydrogen in methanol
T=20°C; 2 h;
参考文献
Lee, Jeewoo; Tran, Phuong-Thao; Hoang, Van-Hai; Thorat, Shivaji A.; Kim, Sung Eun; Ann, Jihyae; Chang, Yu Jin; Nam, Dong Woo; Song, Hyundong; Mook-Jung, Inhee; Lee, Jiyoun
Bioorganic and Medicinal Chemistry, 2013 , vol. 21, # 13 p. 3821 - 3830
