1: With tetra-(n-butyl)ammonium iodide; sodium hydroxide in dichloromethane; water
1 h;
2: With hydrogenchloride; water in dichloromethane
T=20°C; 0.25 h;
参考文献
Vanel, Remi; Berthiol, Florian; Bessieres, Bernard; Einhorn, Cathy; Einhorn, Jacques
Synlett, 2011 , # 9 p. 1293 - 1295
McNamara, Yvonne M.; Cloonan, Suzanne M.; Knox, Andrew J.S.; Keating, John J.; Butler, Stephen G.; Peters, Guenther H.; Meegan, Mary J.; Williams, D. Clive
Bioorganic and Medicinal Chemistry, 2011 , vol. 19, # 3 p. 1328 - 1348