Ladouceur, Gaetan H.; Bullock, William H.; Magnuson, Steven R.; O'Connor, Stephen J.; Smith, Roger A.; Shen, Quanrong; Liu, Qingjie; Su, Ning; Velthuisen, Emil J.; Campbell, Ann-Marie; Ehrlich, Paul P.
Patent: US2003/78258 A1, 2003 ;
1,8-diazabicyclo[5.4.0]undec-7-ene in N,N-dimethyl-formamide T=80°C; 6 h;
参考文献
Armarego, Wilfred L. F.; Taguchi, Hiroyasu; Cotton, Richard G. H.; Battiston, Sandra; Leong, Lillian
European Journal of Medicinal Chemistry, 1987 , vol. 22, p. 283 - 292