1: p-toluidine With hydrogenchloride; sodium nitrite in water T=0 - 5°C; 2: isocyano-acetic acid ethyl ester With sodium acetate in methanol; water T=0 - 20°C;
参考文献
Zibinsky, Mikhail; Fokin, Valery V.
Organic Letters, 2011 , vol. 13, # 18 p. 4870 - 4872
1,8-diazabicyclo[5.4.0]undec-7-ene in N,N-dimethyl-formamide T=80°C; 6 h;
参考文献
Armarego, Wilfred L. F.; Taguchi, Hiroyasu; Cotton, Richard G. H.; Battiston, Sandra; Leong, Lillian
European Journal of Medicinal Chemistry, 1987 , vol. 22, p. 283 - 292