1-氧杂-5-氮杂螺[2.4]庚烷-5-甲酸叔丁酯合成路线 (共 1 条)
反应条件
1: trimethyl-oxo-sulfonium iodide With sodium hydride in dimethyl sulfoxide; mineral oil T=10 - 20°C; 2 h; 2: 3-Oxo-pyrrolidine-1-carboxylic acid tert-butyl ester in dimethyl sulfoxide; mineral oil 3 h;
参考文献
WO2013/138210 A1, ;
Paragraph 0209 ;