1-(6-氯-5H-咪唑并[2,1-b][1,3]噁嗪-3-基)乙酮合成路线 (共 1 条)
反应条件
1: 5-Chloro-pyridin-2-ylamine; N,N-dimethyl-formamide dimethyl acetal 23 h; Heating; 2: 1-bromo-2-propanone in ethanol T=20°C; 18 h; Further stages.;
参考文献
Hayakawa, Masahiko; Kaizawa, Hiroyuki; Kawaguchi, Ken-ichi; Ishikawa, Noriko; Koizumi, Tomonobu; Ohishi, Takahide; Yamano, Mayumi; Okada, Minoru; Ohta, Mitsuaki; Tsukamoto, Shin-ichi; Raynaud, Florence I.; Waterfield, Michael D.; Parker, Peter; Workman, Paul
Bioorganic and Medicinal Chemistry, 2007 , vol. 15, # 1 p. 403 - 412