反应条件
1: potassium carbonate / N,N-dimethyl-formamide / 5 h / 20 °C 2: methanol; sodium methylate / 5 h / 20 °C 3: hydrogen; palladium(II) oxide hydrate / tetrahydrofuran; methanol / 6 h / 20 °C View Scheme
参考文献
Yamasaki, Kazuaki; Hishiki, Ryogo; Kato, Eisuke; Kawabata, Jun
ACS Medicinal Chemistry Letters, 2011 , vol. 2, # 1 p. 17 - 21