2-溴-10h-吲哚并[3,2-b]喹啉合成路线 （共 8 条）
反应条件
in various solvent(s) T=250 - 300°C; Decarboxylation;
参考文献
Caprio, Vittorio; Guyen, Berengere; Opoku-Boahen, Yaw; Mann, John; Gowan, Sharon M.; Kelland, Lloyd M.; Read, Martin A.; Neidle, Stephen
Bioorganic and Medicinal Chemistry Letters, 2000 , vol. 10, # 18 p. 2063 - 2066
反应条件
triethyl phosphite 4 h; Heating;
参考文献
Dutta, Bishnupada; Some, Surajit; Ray, Jayanta K.
Tetrahedron Letters, 2006 , vol. 47, # 3 p. 377 - 379
反应条件
1: aq. KOH / 240 h / 20 °C 2: diphenyl ether / 6 h / 250 °C View Scheme
参考文献
Wright; Addae-Kyereme; Breen; Brown; Cox; Croft; Goekcek; Kendrick; Phillips; Pollet
Journal of Medicinal Chemistry, 2001 , vol. 44, # 19 p. 3187 - 3194
反应条件
1: aq. KOH / 240 h / 20 °C 2: diphenyl ether / 6 h / 250 °C View Scheme
参考文献
Wright; Addae-Kyereme; Breen; Brown; Cox; Croft; Goekcek; Kendrick; Phillips; Pollet
Journal of Medicinal Chemistry, 2001 , vol. 44, # 19 p. 3187 - 3194
反应条件
1: 91 percent / HCl / ethanol / 0 °C 2: 41 percent / 0.08 h / 200 - 250 °C 3: 68 percent / P(OEt)3 / 4 h / Heating View Scheme
参考文献
Dutta, Bishnupada; Some, Surajit; Ray, Jayanta K.
Tetrahedron Letters, 2006 , vol. 47, # 3 p. 377 - 379
反应条件
1: 80 percent / POCl3 / 0 - 80 °C 2: 91 percent / HCl / ethanol / 0 °C 3: 41 percent / 0.08 h / 200 - 250 °C 4: 68 percent / P(OEt)3 / 4 h / Heating View Scheme
参考文献
Dutta, Bishnupada; Some, Surajit; Ray, Jayanta K.
Tetrahedron Letters, 2006 , vol. 47, # 3 p. 377 - 379
反应条件
1: 50 percent / aq. KOH 2: 80 percent / various solvent(s) / 250 - 300 °C View Scheme
参考文献
Caprio, Vittorio; Guyen, Berengere; Opoku-Boahen, Yaw; Mann, John; Gowan, Sharon M.; Kelland, Lloyd M.; Read, Martin A.; Neidle, Stephen
Bioorganic and Medicinal Chemistry Letters, 2000 , vol. 10, # 18 p. 2063 - 2066
反应条件
1: 50 percent / aq. KOH 2: 80 percent / various solvent(s) / 250 - 300 °C View Scheme
参考文献
Caprio, Vittorio; Guyen, Berengere; Opoku-Boahen, Yaw; Mann, John; Gowan, Sharon M.; Kelland, Lloyd M.; Read, Martin A.; Neidle, Stephen
Bioorganic and Medicinal Chemistry Letters, 2000 , vol. 10, # 18 p. 2063 - 2066
