N-叔丁基-3-溴苯磺酰胺合成路线 (共 2 条)
参考文献
Merck Frosst Canada and Co.
Patent: US6316472 B1, 2001 ;
US 6316472 B1
反应条件
caesium carbonate; tris-(dibenzylideneacetone)dipalladium(0); 9,9-dimethyl-4,5-bis(diphenyl-phosphino)xanthene in 1,4-dioxane 3 h; Heating / reflux;
参考文献
TARGEGEN, INC.; TEFFERI, Ayalew
Patent: WO2012/60847 A1, 2012 ;
Location in patent: Page/Page column 42 ;