2-氨基-3-(三氟甲基)苯甲酸合成路线 （共 12 条）
反应条件
1: 50 percent
2: 1.) butyllithium / 1.) THF, hexane, 0 deg C, 20 min, 2.) -70 deg C;
3: 76 percent / 4-N-dimethylaminopyridine / tetrahydrofuran / Ambient temperature
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参考文献
Clemence, Francois; Martret, Odile Le; Collard, Jeannine
Journal of Heterocyclic Chemistry, 1984 , vol. 21, p. 1345 - 1353
反应条件
1: (i) NaNO2, H2SO4, (ii) CuCl, aq. HCl
2: (i) (COCl)2, (ii) NH3
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参考文献
Fuller; Molloy; Day; Roush; Marsh
Journal of medicinal chemistry, 1973 , vol. 16, # 2 p. 101 - 106
