1.1: tBuOK / tetrahydrofuran / 20 °C 1.2: AcOH; TFA / 20 °C 1.3: 74 percent / aq. NH3 / 6 h / Heating 2.1: 84 percent / m-CPBA / CH2Cl2; H2O / 0.67 h / -20 °C View Scheme
参考文献
Majo, Vattoly J.; Prabhakaran, Jaya; Simpson, Norman R.; Van Heertum, Ronald L.; Mann, J. John; Kumar, J. S. Dileep
Bioorganic and Medicinal Chemistry Letters, 2005 , vol. 15, # 19 p. 4268 - 4271