反应条件
1: 99 percent / Cs2CO3 / acetonitrile / 16 h / 20 °C 2: 87 percent / m-chloroperbenzoic acid; p-TsOH / CH2Cl2 / 6 h / Heating 3: NaOCH3; MeOH 4: 100 percent / DMAP; Et3N / dioxane / 16 h / Heating 5: 47 percent / various solvent(s) / 253 °C 6: 34 percent / NaOCH3; MeOH / 16 h / 70 °C 7: Cs2CO3 / acetonitrile / 16 h / 20 °C View Scheme
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 13, # 9 p. 1517 - 1521