2-[(2-羧基苯甲酰基)氨基]戊烷二酸合成路线 (共 1 条)
反应条件
1.1: methyl chloroformate; Et3N / tetrahydrofuran / 0.5 h / 0 °C 1.2: 5.4 percent / tetrahydrofuran / 3 h / 0 - 20 °C 2.1: 99 percent / H2 / Pd/C / dioxane / 2 h / 20 °C View Scheme
参考文献
Nakamura, Takanori; Noguchi, Tomomi; Miyachi, Hiroyuki; Hashimoto, Yuichi
Chemical and Pharmaceutical Bulletin, 2007 , vol. 55, # 4 p. 651 - 654