反应条件
1: 3-Hydroxypyridine-2-carboxylic acid With benzotriazol-1-ol; triethylamine; dicyclohexyl-carbodiimide in N,N-dimethyl-formamide T=20°C; 0.333333 h; 2: 2-amino-thiazole in N,N-dimethyl-formamide T=20°C; 2 h;
参考文献
Luo, Qun-Li; Li, Jing-Ya; Liu, Zhi-Ying; Chen, Ling-Ling; Li, Jia; Qian, Zhen; Shen, Qiang; Li, Yu; Lushington, Gerald H.; Ye, Qi-Zhuang; Nan, Fa-Jun
Journal of Medicinal Chemistry, 2003 , vol. 46, # 13 p. 2631 - 2640