反应条件
1: bis(trichloromethyl) carbonate; 4-[1-(1,4-dioxaspiro[4.5]dec-8-yl)-4-(8-oxa-3-azabicyclo[3.2.1]oct-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-yl]aniline With triethylamine in dichloromethane 2: methylamine in dichloromethane
参考文献
Curran, Kevin J.; Verheijen, Jeroen C.; Kaplan, Joshua; Richard, David J.; Toral-Barza, Lourdes; Hollander, Irwin; Lucas, Judy; Ayral-Kaloustian, Semiramis; Yu, Ker; Zask, Arie
Bioorganic and Medicinal Chemistry Letters, 2010 , vol. 20, # 4 p. 1440 - 1444