1: ZTK-2-124 With n-butyllithium in tetrahydrofuran; hexane T=-78 - 20°C; 1 h; 2: carbon dioxide in tetrahydrofuran; hexane T=-78 - 20°C; 3: With hydrogenchloride in water
Nieland, Nick P.R.; Rennison, David; Broadbear, Jillian H.; Purington, Lauren; Woods, James H.; Traynor, John R.; Lewis, John W.; Husbands, Stephen M.
Journal of Medicinal Chemistry, 2009 , vol. 52, # 21 p. 6926 - 6930