反应条件
1: 2-(3,5-difluorophenyl)acetic acid With (benzotriazo-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; N-ethyl-N,N-diisopropylamine in dichloromethane T=20°C; 1 h; 2: N-(L-alanyl)-(2S)-2-phenylglycine tert-butyl ester With N-ethyl-N,N-diisopropylamine in dichloromethane T=20°C;
参考文献
Pietrancosta, Nicolas; Quelever, Gilles; Laras, Younes; Garino, Cedrik; Burlet, Stephane; Kraus, Jean Louis
Australian Journal of Chemistry, 2005 , vol. 58, # 8 p. 585 - 594