1: in acetone T=-10 - 10°C; 0.75 h; 2: With mercury dichloride in acetone T=-10 - 0°C; 0.25 h; 3: With triethylamine in acetone 1 h; Heating; Further stages.;
参考文献
Park, Soobong; Hayes, Brittany L.; Marankan, Fatima; Mulhearn, Debbie C.; Wanna, Linda; Mesecar, Andrew D.; Santarsiero, Bernard D.; Johnson, Michael E.; Venton, Duane L.
Journal of Medicinal Chemistry, 2003 , vol. 46, # 6 p. 936 - 953