反应条件
1: triethylamine / dichloromethane 2: n-butyllithium; N,N,N',N,-tetramethylethylenediamine / tetrahydrofuran View Scheme
参考文献
F. HOFFMANN-LA ROCHE AG; BISSANTZ, Caterina; DEHMLOW, Henrietta; ERICKSON, Shawn David; KARNACHI, Prabha Saba; KIM, Kyungjin; MARTIN, Rainerm, E.; MATTEI, Patrizio; OBST SANDER, Ulrike; PIETRANICO-COLE, Sherrie Lynn; RICHTER, Hans; ULLMER, Christoph
Patent: WO2012/117000 A1, 2012 ;