反应条件
1: 2-bromo-6-pyridine-carboxylic acid With 1,1'-carbonyldiimidazole in dichloromethane T=20°C; 1 h; 2: N,O-dimethyl-hydroxylamine in dichloromethane T=20°C; 20 h;
参考文献
SMITHKLINE BEECHAM CORPORATION; HAMLETT, Christopher, Charles, Frederick
Patent: WO2004/315 A1, 2003 ;
Location in patent: Page 22 ;
WO 2004/000315 A1