反应条件
1: AlCl3 / 1,2-dichloro-ethane / 2 h / Ambient temperature 2: 1.) Br2, aq. NaOH / 1.) 10 deg C, 2.) dioxane, RT, 1 h 3: LiAlH4 / diethyl ether / 1 h / Heating 4: HCl gas / benzene / 4 h View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 33, # 9 p. 2535 - 2544