反应条件
N,N-dimethyl-aniline; trichlorophosphate
1.) Dowtherm, 230 deg C, 30 min, 2.) 60 deg C, 2 h; Yield given. Multistep reaction. Yields of byproduct given;
参考文献
Abe, Yoshito; Kayakiri, Hiroshi; Satoh, Shigeki; Inoue, Takayuki; Sawada, Yuki; Inamura, Noriaki; Asano, Masayuki; Aramori, Ichiro; Hatori, Chie; Sawai, Hiroe; Oku, Teruo; Tanaka, Hirokazu
Journal of Medicinal Chemistry, 1998 , vol. 41, # 21 p. 4062 - 4079