反应条件
4-(N,N-dimethlyamino)pyridine; potassium carbonate; 1,1'-carbonyldiimidazole in N,N-dimethyl-formamide T=85°C; 4 h;
参考文献
McKie, Jeffrey A.; Bhagwat, Shripad S.; Brady, Helen; Doubleday, Mary; Gayo, Leah; Hickman, Mathew; Jalluri, Ravi K.; Khammungkhune, Sak; Kois, Adam; Mortensen, Deborah; Richard, Normand; Sapienza, John; Shevlin, Graziella; Stein, Bernd; Sutherland, May
Bioorganic and Medicinal Chemistry Letters, 2004 , vol. 14, # 13 p. 3407 - 3410