反应条件
1: 1-t-butoxycarbonyl-4-aminopiperidine With sodium hydride in N,N-dimethyl acetamide T=0°C; 0.25 h; 2: 4-fluoro-nitro-benzene in N,N-dimethyl acetamide T=20°C; Further stages.;
参考文献
Noguchi, Tetsuji; Tanaka, Naoki; Nishimata, Toyoki; Goto, Riki; Hayakawa, Miho; Sugidachi, Atsuhiro; Ogawa, Taketoshi; Asai, Fumitoshi; Ozeki, Tomoko; Fujimoto, Koichi
Chemical and Pharmaceutical Bulletin, 2007 , vol. 55, # 3 p. 393 - 402