1: 58 percent / Cs2CO3; CuI / toluene / Heating
2: 98 percent / aq. NaOH / 0.33 h / 120 °C
3: SOCl2; DMF / CH2Cl2 / 1.5 h / Heating
4: 0.67 g / Et3N / CH2Cl2 / -70 - 20 °C
View Scheme
参考文献
Jarkas, Nachwa; McConathy, Jonathan; Ely, Timothy; Kilts, Clinton D.; Votaw, John; Goodman, Mark M.
Journal of Labelled Compounds and Radiopharmaceuticals, 2001 , vol. 44, p. S204 - S206