7-甲氧基-2,3-二氢-1H-吲哚合成路线 （共 2 条）
反应条件
sodium cyanoborohydride; acetic acid T=0 - 20°C; 1 h;
参考文献
MERCK SHARP and DOHME CORP.; COBURN, Craig, A.; ROSENBLUM, Stuart, B.; KOZLOWSKI, Joseph, A.; SOLL, Richard; WU, Hao; HU, Bin; ZHONG, Bin; WANG, Dahai; SHEN, Changmao; SUN, Fei
Patent: WO2012/122716 A1, 2012 ;
Location in patent: Page/Page column 76 ;
反应条件
1: pyrrolidine / dimethylformamide / 24 h / 130 °C 2: H2 / 10percent Pd/C / 3 h / 2585.7 Torr 3: NaBH3CN / acetic acid / 0.5 h / Ambient temperature View Scheme
参考文献
Gourdoupis; Stamos
Synthetic Communications, 1993 , vol. 23, # 16 p. 2241 - 2249
