反应条件
1: 3-bromophenylacetic acid With N-ethyl-N,N-diisopropylamine; HATU in N,N-dimethyl-formamide T=20°C; 0.25 h; 2: anhydrous cyclopropylamine in N,N-dimethyl-formamide T=20°C;
参考文献
GENELABS TECHNOLOGIES, INC.
Patent: WO2007/70556 A2, 2007 ;
Location in patent: Page/Page column 96 ;