反应条件
1: 67 percent / CuCl 2: 92 percent / POCl3, H2O / dimethylformamide / Vilsmeier reaction 3: ethanol / 1 h / Ambient temperature 4: sodium borohydride / Heating 5: 51 percent / CuCl 6: 89 percent / POCl3, H2O / dimethylformamide / Vilsmeier reaction View Scheme
参考文献
Shawcross, Andrew P.; Stanforth, Stephen P.
Tetrahedron, 1989 , vol. 45, # 22 p. 7063 - 7076