N-苄氧羰基-L-苯丙氨酸，N-羟基琥珀酰亚胺酯合成路线 （共 16 条）
反应条件
dicyclohexyl-carbodiimide in tetrahydrofuran T=0°C; 18 h;
参考文献
Dechert, Anne-Marie R.; MacNamara, James P.; Breevoort, Sarah R.; Hildebrandt, Emily R.; Hembree, Ned W.; Rea, Adam C.; McLain, Duncan E.; Porter, Stephen B.; Schmidt, Walter K.; Dore, Timothy M.
Bioorganic and Medicinal Chemistry, 2010 , vol. 18, # 17 p. 6230 - 6237
反应条件
4-methyl-morpholine in tetrahydrofuran; acetonitrile Ambient temperature;
参考文献
Jaoudai, Mahmoud; Martinez, Jean; Castro, Bertrand
Journal of Organic Chemistry, 1987 , vol. 52, # 12 p. 2364 - 2367
反应条件
1: 85 percent / NaOH 2: 94 percent / dicyclohexylcarbodiimide / dimethylformamide / 5 h / 0 °C View Scheme
参考文献
Tetrahedron Letters, , vol. 29, # 40 p. 5091 - 5094
反应条件
1-hydroxy-pyrrolidine-2,5-dione; dicyclohexyl-carbodiimide in tetrahydrofuran T=0°C; 5 h;
参考文献
Soft Matter, , vol. 7, # 5 p. 2121 - 2126
反应条件
1: 85 percent / NaOH 2: 94 percent / dicyclohexylcarbodiimide / dimethylformamide / 5 h / 0 °C View Scheme
参考文献
Tetrahedron Letters, , vol. 29, # 40 p. 5091 - 5094
反应条件
pyridine in acetonitrile 5 h;
参考文献
Tetrahedron Letters, , vol. 24, # 41 p. 4451 - 4454
反应条件
4-(N,N-dimethlyamino)pyridine in acetonitrile 4 h; Ambient temperature;
参考文献
Synthesis, , # 9 p. 689 - 691
反应条件
pyridine in acetonitrile
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 18, # 20 p. 5559 - 5562
反应条件
sodium tetrahydroborate; acetic acid in 1,4-dioxane; methanol Reduction;
参考文献
Sergeev, Maxim E.; Pronin, Victor B.; Voyushina, Tatiana L.
Synlett, 2005 , # 18 art. no. G24405ST, p. 2802 - 2804
反应条件
1: NaBH4; AcOH / methanol; dioxane 2: MnO2 / CHCl3 / 24 h / 20 °C View Scheme
参考文献
Voyushina, Tatiana L.; Potetinova, Joanna V.; Milgotina, Ekaterina I.; Stepanov, Valentin M.
Bioorganic and Medicinal Chemistry, 1999 , vol. 7, # 12 p. 2953 - 2959
