3-溴-5-二氟甲氧基吡啶合成路线 (共 1 条)
反应条件
potassium hydroxide in water; acetonitrile T=-78 - 80°C; 4 h;
参考文献
INTELLKINE, LLC; INFINITY PHARMACEUTICALS, INC.; CASTRO, Alfredo C.; EVANS, Catherine A.; JANARDANANNAIR, Somarajannair; LESCARBEAU, Andre; LIU, Tao; SNYDER, Daniel A.; TREMBLAY, Martin R.; REN, Pingda; LIU, Yi; LI, Liansheng; CHAN, Katrina
Patent: US2013/53362 A1, 2013 ;
Location in patent: Paragraph 0895; 0896 ;