2-(3-硝基苯基)-2H-1,2,3-噻唑合成路线 （共 2 条）
反应条件
potassium phosphate; N,N-dimethylethylenediamine in N,N-dimethyl-formamide T=110°C; 8 h;
参考文献
GLENMARK PHARMACEUTICALS, S.A.
Patent: WO2009/90548 A2, 2009 ;
Location in patent: Page/Page column 45 ;
WO 2009/090548 A2
反应条件
3,4,5,6-tetramethyl-t-Bu-X-Phos; potassium phosphate; tris-(dibenzylideneacetone)dipalladium(0) in toluene T=120°C; 5 h; Inert atmosphere; regioselective reaction;
参考文献
Ueda, Satoshi; Su, Mingjuan; Buchwald, Stephen L.
Angewandte Chemie - International Edition, 2011 , vol. 50, # 38 p. 8944 - 8947
